Description
WP1066 is a novel inhibitor of JAK2 and STAT3 with IC50 of 2.30 μM and 2.43 μM in HEL cells; shows activity to JAK2, STAT3, STAT5, and ERK1/2 not JAK1 and JAK3.
Storage
2 years -20 centigrade Powder 2 weeks4centigradein DMSO 6 months-80centigradein DMSO
Molecular Formula
C17H14BrN3O
Chemical Name
(S,E)-3-(6-bromopyridin-2-yl)-2-cyano-N-(1-phenylethyl)acrylamide
Solubility
DMSO 72 mg/mL
Water <1 mg/mL
Ethanol <1 mg/mL