Description
Ostarine can selectively inhibit androgen receptor modulator (SARM) with Ki of 3.8 nM. Ostarine at the concentration of 10 nM modulates the transcriptional activity of AR in CV-1 cells cotransfected with a human AR expression vector, a luciferase reporter vector, and a control beta-galactosidase vector, with 94%-100% relative activity of the transcriptional activation observed for 1 nM DHT.
Alias
GTx-024, MK-2866, Enobosarm, S-22
Storage
2 years at -20centigrade Powder
Synonyms
GTx-024, MK-2866, Enobosarm, S-22
Molecular Formula
C19H14F3N3O3
Chemical Name
(S)-N-(4-cyano-3-(trifluoromethyl)phenyl)-3-(4-cyanophenoxy)-2-hydroxy-2-methylpropanamide
Solubility
DMSO 78 mg/mL, Water
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