Products
Online Inquiry
Our Products Cannot Be Used As Medicines Directly For Personal Use.
Welcome! For price inquiries, please feel free to contact us through the form on the left side. We will get back to you as soon as possible.
GF-109203X
Cat No.
CEI-0963
Description
Potent and selective protein kinase C inhibitor with specificity for the alpha and beta1 isotypes. IC50=0.0084, 0.018, 0.210, 0.132 and 0.58 uM for alpha, beta1, delta, epsilon, and zeta respectively. An extremely useful tool for assessing the involvement of PKC in various signaling pathways.
Abbr
GF-109203X (PRRT2)
Alias
1. 2-[1-(3-Dimethylaminopropyl)-1H-indol-3-yl]-3-(1H-indol-3-yl) maleimide 2. Bisindolylmaleimide I
Appearance
Red/orange powder
Product Overview
PKC inhibitor
CAS No.
133052-90-1
Molecular Weight
412.5
Purity
98% (TLC); NMR (Conforms)
Synonyms
1. 2-[1-(3-Dimethylaminopropyl)-1H-indol-3-yl]-3-(1H-indol-3-yl) maleimide 2. Bisindolylmaleimide I
Targets
PKC
Molecular Formula
C25H24N4O2
Solubility
Soluble in dimethyl formamide or DMSO (10mg/ml, warm to 40oC)
Download
Download Datasheet