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EZH2 Inhibitor, EPZ005687

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Cat No.

CEI-0475

Description

A potent and selective inhibitor of histone lysine N-methyltransferase EZH2 (Ki = 24 nM). It displays more than 500-fold selectivity against 15 other protein methyltransferases and has 50-fold selectivity against the closely related enzyme, EZH1.

Appearance

White to off-white solid

Product Overview

A potent EZH2 inhibitor

CAS No.

1396772-26-1

Molecular Weight

475.6

Purity

>98% by HPLC

Storage

+4 centigrade

Targets

EZH2

Molecular Formula

C 32 H 37 N 6 O 3

Chemical Name

1-Cyclopentyl-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-6-(4-(morpholinomethyl)phenyl)-1H-indazole-4-carboxamide

Solubility

DMSO (10 mg/ml)

Shipping Conditions

Gel pack