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EZH2 Inhibitor, EPZ005687
Cat No.
CEI-0475
Description
A potent and selective inhibitor of histone lysine N-methyltransferase EZH2 (Ki = 24 nM). It displays more than 500-fold selectivity against 15 other protein methyltransferases and has 50-fold selectivity against the closely related enzyme, EZH1.
Appearance
White to off-white solid
Product Overview
A potent EZH2 inhibitor
CAS No.
1396772-26-1
Molecular Weight
475.6
Purity
>98% by HPLC
Storage
+4 centigrade
Targets
EZH2
Molecular Formula
C 32 H 37 N 6 O 3
Chemical Name
1-Cyclopentyl-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-6-(4-(morpholinomethyl)phenyl)-1H-indazole-4-carboxamide
Solubility
DMSO (10 mg/ml)
Shipping Conditions
Gel pack
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