Description
Cell-permeable. A potent and specific protein arginine N-methyltransferase (PRMTs) inhibitor (IC50 = 8.8 µM for human PRMT1 and 3.0 µM for yeast Hmt1p ). Does not compete for the AdoMet (S-adenosyl-L-methionine; SAM) binding site. Also acts as a HIV-1 RT polymerase inhibitor (IC50 = 5.0 µM).
Alias
Arginine N-methyltransferase inhibitor-1
Product Overview
A potent and specific protein arginine N-methyltransferase (PRMTs) inhibitor
Synonyms
Arginine N-methyltransferase inhibitor-1
Molecular Formula
C₂₁H₁₂N₂O₉S₂Na₄
Shipping Conditions
Gel pack
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