Products
Online Inquiry
Our Products Cannot Be Used As Medicines Directly For Personal Use.
Welcome! For price inquiries, please feel free to contact us through the form on the left side. We will get back to you as soon as possible.
(R)-MG132
Cat No.
CEI-1002
Description
(R)-MG132 is a potent, cell permeable and reversible inhibitor of proteasomes. It can inhibit proteasome activity in lysates of J558L multiple myeloma cells and EMT6 breast cancer cells. In comparison to (S)-MG132, the (R)-MG132 stereoisomer is a more effective inhibitor of chymotrypsin-like (ChTL), trypsin-like (TL), and peptidylglutamyl peptide hydrolyzing proteasome (PGPH) activities.
Abbr
(R)-MG132(ChTL, TLa, PGPH)
Appearance
A crystalline solid.
CAS No.
1211877-36-9
Molecular Weight
475.6
Purity
>98%
Storage
Store at or below -20 centigrade for up to two years.
Targets
ChTL, TLa, PGPH
IC50
0.22 µM, 34.4 µM, 2.95 µM
Molecular Formula
C26H41N3O5
Download
Download Datasheet