Description
TG100713 is a pan-PI3K inhibitor against PI3Kγ, PI3Kδ, PI3Kα and PI3Kβ with IC50 of 50 nM, 24 nM, 165 nM and 215 nM, respectively.
Storage
2 years -20 centigrade Powder; 2 weeks 4 centigrade in DMSO; 6 months -80 centigrade in DMSO.
Targets
PI3Kγ, PI3Kδ, PI3Kα, PI3Kβ
IC50
50 nM; 24 nM; 165 nM; 215 nM
Molecular Formula
C12H10N6
Chemical Name
Phenol, 3-(2,4-diamino-6-pteridinyl)-
Solubility
DMSO 2 mg/mL; Water <1 mg/mL; Ethanol <1 mg/mL
In vitro
TG 100713 also strongly inhibits EC proliferation.